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5DKN

Crystal Structure of Calcium-loaded S100B bound to SBi4225

Summary for 5DKN
Entry DOI10.2210/pdb5dkn/pdb
Related5DKQ 5DKR
DescriptorProtein S100-B, CALCIUM ION, 2,2'-[heptane-1,7-diylbis(oxybenzene-4,1-diyl)]bis(1H-imidazole), ... (4 entities in total)
Functional Keywordsmalignant melanoma, calcium binding, covalent inhibitor, metal binding protein-inhibitor complex, metal binding protein/inhibitor
Biological sourceBos taurus (Bovine)
Total number of polymer chains1
Total formula weight11178.65
Authors
Primary citationCavalier, M.C.,Ansari, M.I.,Pierce, A.D.,Wilder, P.T.,McKnight, L.E.,Raman, E.P.,Neau, D.B.,Bezawada, P.,Alasady, M.J.,Charpentier, T.H.,Varney, K.M.,Toth, E.A.,MacKerell, A.D.,Coop, A.,Weber, D.J.
Small Molecule Inhibitors of Ca(2+)-S100B Reveal Two Protein Conformations.
J.Med.Chem., 59:592-608, 2016
Cited by
PubMed: 26727270
DOI: 10.1021/acs.jmedchem.5b01369
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.528 Å)
Structure validation

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