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5CS2

Crystal structure of Plasmodium falciparum diadenosine triphosphate hydrolase in complex with Cyclomarin A

Summary for 5CS2
Entry DOI10.2210/pdb5cs2/pdb
DescriptorHistidine triad protein, Cyclomarin A, CHLORIDE ION, ... (4 entities in total)
Functional Keywordscyclomarin a, diadenosine triphosphate hydrolase, anti-plasmodial activity, malaria, plasmodium falciparum, hydrolase
Biological sourcePlasmodium falciparum 3D7
More
Total number of polymer chains2
Total formula weight24744.58
Authors
Ostermann, N.,Schmitt, E.,Gerhartz, B.,Hinniger, A.,Delmas, C. (deposition date: 2015-07-23, release date: 2015-10-28, Last modification date: 2024-01-10)
Primary citationBurstner, N.,Roggo, S.,Ostermann, N.,Blank, J.,Delmas, C.,Freuler, F.,Gerhartz, B.,Hinniger, A.,Hoepfner, D.,Liechty, B.,Mihalic, M.,Murphy, J.,Pistorius, D.,Rottmann, M.,Thomas, J.R.,Schirle, M.,Schmitt, E.K.
Gift from Nature: Cyclomarin A Kills Mycobacteria and Malaria Parasites by Distinct Modes of Action.
Chembiochem, 16:2433-2436, 2015
Cited by
PubMed: 26472355
DOI: 10.1002/cbic.201500472
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.65 Å)
Structure validation

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