5C89

Crystal structure of the human BRPF1 bromodomain in complex with 917

Summary for 5C89

• Entry DOI: 10.2210/pdb5c89/pdb
• Related: 5C7N 5C85 5C87
• Descriptor: Peregrin, 1-ethyl-8-methoxy-5-methyl[1,2,4]triazolo[4,3-a]quinoline (3 entities in total)
• Functional Keywords: bromodomain and phd finger-containing protein 1(brpf1), monocytic leukemia zinc-finger (moz), inhibitor, dna binding protein
• Biological source: Homo sapiens (Human)
• Cellular location: Nucleus : P55201
• Total number of polymer chains: 1
• Total formula weight: 13944.99

Authors

Zhu, J.,Wiedmer, L.,Caflisch, A. (deposition date: 2015-06-25, release date: 2016-07-13, Last modification date: 2024-01-10)

• Primary citation: Zhu, J.,Caflisch, A.; Crystal structure of the human BRPF1 bromodomain in complex with 917; To Be Published,

Experimental method

X-RAY DIFFRACTION (1.65 Å)