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5C67

Human Mesotrypsin in complex with amyloid precursor protein inhibitor variant APPI-M17G/I18F/F34V

Summary for 5C67
Entry DOI10.2210/pdb5c67/pdb
DescriptorTrypsin-3, Amyloid beta A4 protein (3 entities in total)
Functional Keywordsappi, kunitz domain, trypsin, hyrdolase-hydrolase inhibitor complex, hyrdolase/hydrolase inhibitor
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains4
Total formula weight66784.71
Authors
Kayode, O.,Sankaran, B.,Radisky, E.S. (deposition date: 2015-06-22, release date: 2016-05-04, Last modification date: 2023-09-27)
Primary citationCohen, I.,Kayode, O.,Hockla, A.,Sankaran, B.,Radisky, D.C.,Radisky, E.S.,Papo, N.
Combinatorial protein engineering of proteolytically resistant mesotrypsin inhibitors as candidates for cancer therapy.
Biochem.J., 473:1329-1341, 2016
Cited by
PubMed: 26957636
DOI: 10.1042/BJ20151410
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.83 Å)
Structure validation

217705

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