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5B6G

Protein-protein interaction

Summary for 5B6G
Entry DOI10.2210/pdb5b6g/pdb
DescriptorAdenomatous polyposis coli protein, PHQ-ALA-GLY-GLU-ALA-XYC-TYR-GLU, SULFATE ION, ... (5 entities in total)
Functional Keywordsapc, asef, colon cancer, drug discovery, protein binding-inhibitor complex, protein binding/inhibitor
Biological sourceHomo sapiens (Human)
More
Total number of polymer chains2
Total formula weight40384.81
Authors
Zhao, Y.,Jiang, H.,Yang, X.,Jiang, F.,Song, K.,Zhang, J. (deposition date: 2016-05-27, release date: 2017-05-31, Last modification date: 2023-11-08)
Primary citationJiang, H.,Deng, R.,Yang, X.,Shang, J.,Lu, S.,Zhao, Y.,Song, K.,Liu, X.,Zhang, Q.,Chen, Y.,Chinn, Y.E.,Wu, G.,Li, J.,Chen, G.,Yu, J.,Zhang, J.
Peptidomimetic inhibitors of APC-Asef interaction block colorectal cancer migration.
Nat. Chem. Biol., 13:994-1001, 2017
Cited by
PubMed: 28759015
DOI: 10.1038/nchembio.2442
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.99 Å)
Structure validation

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