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5A14

Human CDK2 with type II inhibitor

Summary for 5A14
Entry DOI10.2210/pdb5a14/pdb
DescriptorCYCLIN-DEPENDENT KINASE 2, 1-[4-(2-azanylpyrimidin-4-yl)oxyphenyl]-3-[4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl]urea (3 entities in total)
Functional Keywordstransferase, cdk2, cyclin, kinase, type ii, inhibitor
Biological sourceHOMO SAPIENS (HUMAN)
Total number of polymer chains1
Total formula weight35005.54
Authors
Primary citationAlexander, L.T.,Mobitz, H.,Drueckes, P.,Savitsky, P.,Fedorov, O.,Elkins, J.M.,Deane, C.M.,Cowan-Jacob, S.W.,Knapp, S.
Type II Inhibitors Targeting Cdk2.
Acs Chem.Biol., 10:2116-, 2015
Cited by
PubMed: 26158339
DOI: 10.1021/ACSCHEMBIO.5B00398
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2 Å)
Structure validation

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