5TS8
Z. MAYS CK2 KINASE ALPHA SUBUNIT IN COMPLEX WITH THE ATP-COMPETITIVE INHIBITOR 5,6-DIBROMOBENZOTRIAZOLE
Summary for 5TS8
Entry DOI | 10.2210/pdb5ts8/pdb |
Related | 1DAW 1J91 1P5E 2OXY 4KWP 4RKL |
Descriptor | Protein kinase CK2 catalytic subunit CK2 alpha-3, 5,6-DIBROMOBENZOTRIAZOLE, L(+)-TARTARIC ACID, ... (10 entities in total) |
Functional Keywords | ck2, casein kinase 2, inhibitor, bromo-benzotriazole, transferase-transferase inhibitor complex, halogen bond, transferase/transferase inhibitor |
Biological source | Zea mays |
Total number of polymer chains | 1 |
Total formula weight | 41490.89 |
Authors | Winiewska, M.,Kucinska, K.,Czapinska, H.,Piasecka, A.,Bochtler, M.,Poznanski, J. (deposition date: 2016-10-28, release date: 2018-01-17, Last modification date: 2024-01-17) |
Primary citation | Winiewska, M.,Kucinska, K.,Czapinska, H.,Piasecka, A.,Bochtler, M.,Poznanski, J. STRUCTURAL AND THERMODYNAMIC ANALYSIS OF 5,6-DIBROMOBENZOTRIAZOLE BINDING TO CASEIN KINASE 2 ALPHA To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.45 Å) |
Structure validation
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