5LBT
Structure of the human quinone reductase 2 (NQO2) in complex with imiquimod
Summary for 5LBT
Entry DOI | 10.2210/pdb5lbt/pdb |
Descriptor | Ribosyldihydronicotinamide dehydrogenase [quinone], ZINC ION, FLAVIN-ADENINE DINUCLEOTIDE, ... (6 entities in total) |
Functional Keywords | quinone reductase 2 ribosyldihydronicotinamide dehydrogenase, oxidoreductase |
Biological source | Homo sapiens (Human) |
Cellular location | Cytoplasm: P16083 |
Total number of polymer chains | 2 |
Total formula weight | 56502.12 |
Authors | Schneider, S.,Gross, O. (deposition date: 2016-06-17, release date: 2016-07-27, Last modification date: 2024-01-10) |
Primary citation | Gross, C.,Mishra, R.,Schneider, K.,Medard, G.,Wettmarshausen, J.,Dittlein, D.,Gorka, O.,Koenig, P.-A.,Fromm, S.,Magnani, G.,Cikovic, T.,Hartjes, L.,Smollich, J.,Robertson, A.,Cooper, M.,Schmidt-Supprian, M.,Schuster, M.,Schroder, K.,Broz, P.,Traidl-Hoffmann, C.,Kuester, B.,Ruland, J.,Schneider, S.,Perocchi, F.,Gross, O. Imiquimod Inhibits Mitochondrial Complex I and Induces K+ efflux-independent Nlrp3 Inflammasome Activation via Nek7 To Be Published, |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
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