5I40
BRD9 in complex with Cpd1 (6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one)
Summary for 5I40
Entry DOI | 10.2210/pdb5i40/pdb |
Descriptor | Bromodomain-containing protein 9, 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, ... (5 entities in total) |
Functional Keywords | bromodomain inhibitor epigenetics structure-based drug design, rna binding protein |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 12359.48 |
Authors | Murray, J.M. (deposition date: 2016-02-11, release date: 2016-10-12, Last modification date: 2024-03-06) |
Primary citation | Crawford, T.D.,Tsui, V.,Flynn, E.M.,Wang, S.,Taylor, A.M.,Cote, A.,Audia, J.E.,Beresini, M.H.,Burdick, D.J.,Cummings, R.,Dakin, L.A.,Duplessis, M.,Good, A.C.,Hewitt, M.C.,Huang, H.R.,Jayaram, H.,Kiefer, J.R.,Jiang, Y.,Murray, J.,Nasveschuk, C.G.,Pardo, E.,Poy, F.,Romero, F.A.,Tang, Y.,Wang, J.,Xu, Z.,Zawadzke, L.E.,Zhu, X.,Albrecht, B.K.,Magnuson, S.R.,Bellon, S.,Cochran, A.G. Diving into the Water: Inducible Binding Conformations for BRD4, TAF1(2), BRD9, and CECR2 Bromodomains. J.Med.Chem., 59:5391-5402, 2016 Cited by PubMed: 27219867DOI: 10.1021/acs.jmedchem.6b00264 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.0402 Å) |
Structure validation
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