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5I40

BRD9 in complex with Cpd1 (6-methyl-1,6-dihydro-7H-pyrrolo[2,3-c]pyridin-7-one)

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue EDO A 201
ChainResidue
ALYS71
AVAL82
ATHR83
ALYS86
AHOH307

site_idAC2
Number of Residues7
Detailsbinding site for residue EDO A 202
ChainResidue
AILE53
A67N206
AHOH331
AGLY43
APHE44
AALA46
APHE47

site_idAC3
Number of Residues8
Detailsbinding site for residue EDO A 203
ChainResidue
AGLN37
AALA46
APHE47
AGLY68
APHE118
AHOH314
AHOH353
AHOH362

site_idAC4
Number of Residues5
Detailsbinding site for residue EDO A 204
ChainResidue
ATHR50
AASP51
AHOH336
AHOH384
AHOH392

site_idAC5
Number of Residues7
Detailsbinding site for residue PEG A 205
ChainResidue
APRO48
ATHR69
AASP72
AHOH307
AHOH362
AHOH412
AHOH415

site_idAC6
Number of Residues9
Detailsbinding site for residue 67N A 206
ChainResidue
APHE44
APHE45
AVAL49
AILE53
AALA54
AASN100
ATYR106
AEDO202
AHOH306

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding => ECO:0000269|PubMed:26365797
ChainResidueDetails
AILE53
ATYR106

223166

PDB entries from 2024-07-31

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