4YUQ
CDPK1 from Eimeria tenella in complex with inhibitor UW1354
Summary for 4YUQ
Entry DOI | 10.2210/pdb4yuq/pdb |
Related | 4ysj 4ysm |
Descriptor | Calmodulin-like domain protein kinase, CALCIUM ION, 1-cyclopentyl-3-(1H-pyrrolo[2,3-b]pyridin-5-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine (3 entities in total) |
Functional Keywords | serine/threonine protein kinase, transferase, calcium-binding, atp-binding, bumped kinase inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Eimeria tenella (Coccidian parasite) |
Total number of polymer chains | 2 |
Total formula weight | 112296.36 |
Authors | Merritt, E.A. (deposition date: 2015-03-19, release date: 2016-04-06, Last modification date: 2023-09-27) |
Primary citation | Ojo, K.K.,Vidadala, R.,Maly, D.J.,Van Voorhis, W.C.,Merritt, E.A. CDPK is a druggable target in the apicomplexan parasite Eimeria to be published, |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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