4YC0
Crystal structure of ADP-ribosyltransferase Vis in complex with M6 Inhibitor
Summary for 4YC0
Entry DOI | 10.2210/pdb4yc0/pdb |
Descriptor | Putative NAD(+)--arginine ADP-ribosyltransferase Vis, 2-(4-oxidanylidene-3~{H}-phthalazin-1-yl)ethanoic acid (3 entities in total) |
Functional Keywords | inhibitor, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Vibrio splendidus |
Total number of polymer chains | 1 |
Total formula weight | 27241.23 |
Authors | Ravulapalli, R.,Merrill, A.R. (deposition date: 2015-02-19, release date: 2015-11-18, Last modification date: 2023-09-27) |
Primary citation | Ravulapalli, R.,Lugo, M.R.,Pfoh, R.,Visschedyk, D.,Poole, A.,Fieldhouse, R.J.,Pai, E.F.,Merrill, A.R. Characterization of Vis Toxin, a Novel ADP-Ribosyltransferase from Vibrio splendidus. Biochemistry, 54:5920-5936, 2015 Cited by PubMed: 26352925DOI: 10.1021/acs.biochem.5b00921 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5 Å) |
Structure validation
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