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4YC0

Crystal structure of ADP-ribosyltransferase Vis in complex with M6 Inhibitor

Summary for 4YC0
Entry DOI10.2210/pdb4yc0/pdb
DescriptorPutative NAD(+)--arginine ADP-ribosyltransferase Vis, 2-(4-oxidanylidene-3~{H}-phthalazin-1-yl)ethanoic acid (3 entities in total)
Functional Keywordsinhibitor, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceVibrio splendidus
Total number of polymer chains1
Total formula weight27241.23
Authors
Ravulapalli, R.,Merrill, A.R. (deposition date: 2015-02-19, release date: 2015-11-18, Last modification date: 2023-09-27)
Primary citationRavulapalli, R.,Lugo, M.R.,Pfoh, R.,Visschedyk, D.,Poole, A.,Fieldhouse, R.J.,Pai, E.F.,Merrill, A.R.
Characterization of Vis Toxin, a Novel ADP-Ribosyltransferase from Vibrio splendidus.
Biochemistry, 54:5920-5936, 2015
Cited by
PubMed: 26352925
DOI: 10.1021/acs.biochem.5b00921
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.5 Å)
Structure validation

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