4XJM
Crystal structure of 7,8-diaminopelargonic acid synthase (BioA) from Mycobacterium tuberculosis, complexed with a HTS lead compound
Summary for 4XJM
Entry DOI | 10.2210/pdb4xjm/pdb |
Related | 4XJL 4XJO 4XJP |
Descriptor | Adenosylmethionine-8-amino-7-oxononanoate aminotransferase, 3-{1-[(5-acetylthiophen-2-yl)carbonyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide, PYRIDOXAL-5'-PHOSPHATE, ... (4 entities in total) |
Functional Keywords | inhibitor complex transaminase plp, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Mycobacterium tuberculosis (strain ATCC 25618 / H37Rv) |
Total number of polymer chains | 2 |
Total formula weight | 98396.36 |
Authors | Finzel, B.C.,Dai, R. (deposition date: 2015-01-08, release date: 2016-01-20, Last modification date: 2023-09-27) |
Primary citation | Finzel, B.C.,Dai, R. Fragment based inhibitor design of Mycobacterium tuberculosis BioA (http://hdl.handle.net/11299/171084) Thesis, University of Minnesota, 2015 |
Experimental method | X-RAY DIFFRACTION (1.6 Å) |
Structure validation
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