4XI2
Crystal Structure of an auto-inhibited form of Bruton's Tryrosine Kinase
Summary for 4XI2
Entry DOI | 10.2210/pdb4xi2/pdb |
Descriptor | Tyrosine-protein kinase BTK, GOLD ION (2 entities in total) |
Functional Keywords | kinase, phosphorylation, auto-inhibited, b-cell development, x-linked agammaglobulinemia, transferase |
Biological source | Mus musculus (Mouse) |
Cellular location | Cytoplasm : P35991 |
Total number of polymer chains | 1 |
Total formula weight | 52192.75 |
Authors | Vogan, E.M.,Harrison, S.C. (deposition date: 2015-01-06, release date: 2015-02-25, Last modification date: 2024-02-28) |
Primary citation | Wang, Q.,Vogan, E.M.,Nocka, L.M.,Rosen, C.E.,Zorn, J.A.,Harrison, S.C.,Kuriyan, J. Autoinhibition of Bruton's tyrosine kinase (Btk) and activation by soluble inositol hexakisphosphate. Elife, 4:-, 2015 Cited by PubMed: 25699547DOI: 10.7554/eLife.06074 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.6 Å) |
Structure validation
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