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4WG5

Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with inhibitor UW1647

Summary for 4WG5
Entry DOI10.2210/pdb4wg5/pdb
Related4WG3 4WG5
DescriptorCalmodulin-domain protein kinase 1, 5-amino-3-[7-(cyclobutyloxy)quinolin-3-yl]-1-cyclohexyl-1H-pyrazole-4-carboxamide (3 entities in total)
Functional Keywordsserine/threonine protein kinase, transferase, calcium-binding, atp-binding, bumped kinase inhibitor, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceToxoplasma gondii
Total number of polymer chains1
Total formula weight55632.41
Authors
Merritt, E.A. (deposition date: 2014-09-17, release date: 2014-10-15, Last modification date: 2023-12-27)
Primary citationMerritt, E.A.,Maly, D.J.,Ojo, K.K.,Zhang, Z.,Fan, E.,Van Voorhis, W.C.
Calcium-Dependent Protein Kinase 1 from Toxoplasma gondii (TgCDPK1) in complex with inhibitor UW1647
to be published,
Experimental method
X-RAY DIFFRACTION (2.3 Å)
Structure validation

217705

PDB entries from 2024-03-27

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