4WAE
Phosphatidylinositol 4-kinase III beta crystallized with ATP
Summary for 4WAE
Entry DOI | 10.2210/pdb4wae/pdb |
Descriptor | Phosphatidylinositol 4-kinase beta,Phosphatidylinositol 4-kinase beta, ADENOSINE-5'-TRIPHOSPHATE (2 entities in total) |
Functional Keywords | transferase |
Biological source | Homo sapiens (Human) More |
Cellular location | Endomembrane system: Q9UBF8 |
Total number of polymer chains | 1 |
Total formula weight | 65771.95 |
Authors | Chalupska, D.,Boura, E. (deposition date: 2014-08-29, release date: 2015-05-20, Last modification date: 2024-01-10) |
Primary citation | Mejdrova, I.,Chalupska, D.,Kogler, M.,Sala, M.,Plackova, P.,Baumlova, A.,Hrebabecky, H.,Prochazkova, E.,Dejmek, M.,Guillon, R.,Strunin, D.,Weber, J.,Lee, G.,Birkus, G.,Mertlikova-Kaiserova, H.,Boura, E.,Nencka, R. Highly Selective Phosphatidylinositol 4-Kinase III beta Inhibitors and Structural Insight into Their Mode of Action. J.Med.Chem., 58:3767-3793, 2015 Cited by PubMed: 25897704DOI: 10.1021/acs.jmedchem.5b00499 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.318 Å) |
Structure validation
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