4TND
Crystal Structure of G Protein-Coupled Receptor Kinase 5 in Complex with AMP-PNP
Summary for 4TND
Entry DOI | 10.2210/pdb4tnd/pdb |
Related | 4TNB |
Descriptor | G protein-coupled receptor kinase 5, PHOSPHOAMINOPHOSPHONIC ACID-ADENYLATE ESTER, MAGNESIUM ION, ... (4 entities in total) |
Functional Keywords | grk5-(5-adenylylimidodiphosphate) complex, grk5-(amp-pnp) complex, gpcr kinase, kinase, gpcr kinase 5, signaling protein |
Biological source | Homo sapiens (Human) |
Cellular location | Cytoplasm: P34947 |
Total number of polymer chains | 1 |
Total formula weight | 68473.17 |
Authors | Bhardwaj, A.,Komolov, K.E.,Benovic, J.L. (deposition date: 2014-06-04, release date: 2015-06-10, Last modification date: 2023-09-27) |
Primary citation | Komolov, K.E.,Bhardwaj, A.,Benovic, J.L. Atomic Structure of G Protein-Coupled Receptor Kinase 5 (GRK5) Reveals Distinct Structural Features Novel for GRKs. J.Biol.Chem., 2015 Cited by PubMed: 26032409DOI: 10.1074/jbc.M115.647297 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.802 Å) |
Structure validation
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