4OLI
The pseudokinase/kinase protein from JAK-family member TYK2
Summary for 4OLI
Entry DOI | 10.2210/pdb4oli/pdb |
Descriptor | Non-receptor tyrosine-protein kinase TYK2, 2-chloro-N-{2-[(cyclopropylcarbonyl)amino]pyridin-4-yl}benzamide (3 entities in total) |
Functional Keywords | protein kinase, phospho-transfer, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 1 |
Total formula weight | 73935.73 |
Authors | Eigenbrot, C.,Ultsch, M.,Wallweber, H. (deposition date: 2014-01-23, release date: 2014-05-28, Last modification date: 2023-09-20) |
Primary citation | Lupardus, P.J.,Ultsch, M.,Wallweber, H.,Bir Kohli, P.,Johnson, A.R.,Eigenbrot, C. Structure of the pseudokinase-kinase domains from protein kinase TYK2 reveals a mechanism for Janus kinase (JAK) autoinhibition. Proc.Natl.Acad.Sci.USA, 111:8025-8030, 2014 Cited by PubMed: 24843152DOI: 10.1073/pnas.1401180111 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.8 Å) |
Structure validation
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