4O9R
Human Smoothened Receptor structure in complex with cyclopamine
4O9R の概要
エントリーDOI | 10.2210/pdb4o9r/pdb |
分子名称 | Smoothened homolog/Soluble cytochrome b562 chimeric protein, Cyclopamine (2 entities in total) |
機能のキーワード | serial femtosecond crystallography, human smo receptor, cyclopamine, novel protein engineering, gpcr network, psi-biology, free electron laser, structural genomics, membrane protein, xfel, lcp, room temperature structure, gpcr, membrane, signaling protein |
由来する生物種 | Homo sapiens 詳細 |
細胞内の位置 | Membrane ; Multi-pass membrane protein : Q99835 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 52806.82 |
構造登録者 | Wang, C.,Weierstall, U.,James, D.,White, T.A.,Wang, D.,Liu, W.,Spence, J.C.H.,Doak, R.B.,Nelson, G.,Fromme, P.,Fromme, R.,Grotjohann, I.,Kupitz, C.,Zatsepin, N.A.,Liu, H.,Basu, S.,Wacker, D.,Han, G.W.,Katritch, V.,Boutet, S.,Messerschmidt, M.,Willams, G.J.,Koglin, J.E.,Seibert, M.M.,Klinker, M.,Gati, C.,Shoeman, R.L.,Barty, A.,Chapman, H.N.,Kirian, R.A.,Beyerlein, K.R.,Stevens, R.C.,Li, D.,Shah, S.T.A.,Howe, N.,Caffrey, M.,Cherezov, V.,GPCR Network (GPCR) (登録日: 2014-01-02, 公開日: 2014-03-05, 最終更新日: 2023-09-20) |
主引用文献 | Weierstall, U.,James, D.,Wang, C.,White, T.A.,Wang, D.,Liu, W.,Spence, J.C.,Bruce Doak, R.,Nelson, G.,Fromme, P.,Fromme, R.,Grotjohann, I.,Kupitz, C.,Zatsepin, N.A.,Liu, H.,Basu, S.,Wacker, D.,Han, G.W.,Katritch, V.,Boutet, S.,Messerschmidt, M.,Williams, G.J.,Koglin, J.E.,Marvin Seibert, M.,Klinker, M.,Gati, C.,Shoeman, R.L.,Barty, A.,Chapman, H.N.,Kirian, R.A.,Beyerlein, K.R.,Stevens, R.C.,Li, D.,Shah, S.T.,Howe, N.,Caffrey, M.,Cherezov, V. Lipidic cubic phase injector facilitates membrane protein serial femtosecond crystallography. Nat Commun, 5:3309-3309, 2014 Cited by PubMed: 24525480DOI: 10.1038/ncomms4309 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (3.204 Å) |
構造検証レポート
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