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4M2X

Mycobacterium tuberculosis dihydrofolate reductase complexed with trimetrexate (TMQ)

Summary for 4M2X
Entry DOI10.2210/pdb4m2x/pdb
DescriptorDihydrofolate reductase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, TRIMETREXATE, ... (6 entities in total)
Functional Keywordsstructural genomics, tb structural genomics consortium, tbsgc, reductase, nadph binding, hydride transfer, oxidoreductase-oxidoreductase inhibitor complex, oxidoreductase/oxidoreductase inhibitor
Biological sourceMycobacterium tuberculosis
Total number of polymer chains4
Total formula weight77630.41
Authors
Jung, H.,Sacchettini, J.C.,TB Structural Genomics Consortium (TBSGC) (deposition date: 2013-08-05, release date: 2014-11-12, Last modification date: 2024-02-28)
Primary citationJung, H.,Sacchettini, J.C.
Selective inhibitors for dihydrofolate reductase from mycobacterium tuberculosis
To be Published,
Experimental method
X-RAY DIFFRACTION (2.26 Å)
Structure validation

217705

数据于2024-03-27公开中

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