4LH4
Dual inhibition of HIV-1 replication by Integrase-LEDGF allosteric inhibitors is predominant at post-integration stage during virus production rather than at integration
Summary for 4LH4
Entry DOI | 10.2210/pdb4lh4/pdb |
Related | 1BHL 4LH5 |
Descriptor | Integrase, MAGNESIUM ION (3 entities in total) |
Functional Keywords | integrase, transferase |
Biological source | Human immunodeficiency virus 1 |
Total number of polymer chains | 1 |
Total formula weight | 20163.95 |
Authors | |
Primary citation | Le Rouzic, E.,Bonnard, D.,Chasset, S.,Bruneau, J.M.,Chevreuil, F.,Le Strat, F.,Nguyen, J.,Beauvoir, R.,Amadori, C.,Brias, J.,Vomscheid, S.,Eiler, S.,Levy, N.,Delelis, O.,Deprez, E.,Saib, A.,Zamborlini, A.,Emiliani, S.,Ruff, M.,Ledoussal, B.,Moreau, F.,Benarous, R. Dual inhibition of HIV-1 replication by integrase-LEDGF allosteric inhibitors is predominant at the post-integration stage. Retrovirology, 10:144-144, 2013 Cited by PubMed: 24261564DOI: 10.1186/1742-4690-10-144 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.8 Å) |
Structure validation
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