4K4O
The DNA Gyrase B ATP binding domain of Enterococcus faecalis in complex with a small molecule inhibitor
Summary for 4K4O
Entry DOI | 10.2210/pdb4k4o/pdb |
Descriptor | DNA gyrase subunit B, 6-fluoro-4-[(3aR,6aR)-hexahydropyrrolo[3,4-b]pyrrol-5(1H)-yl]-N-methyl-2-[(2-methylpyrimidin-5-yl)oxy]-9H-pyrimido[4,5-b]indol-8-amine, TERTIARY-BUTYL ALCOHOL, ... (4 entities in total) |
Functional Keywords | atp-binding, nucleotide-binding, topoisomerase, atp-binding domain, isomerase-isomerase inhibitor complex, cytosol, isomerase/isomerase inhibitor |
Biological source | Enterococcus faecalis |
Cellular location | Cytoplasm (By similarity): Q839Z1 |
Total number of polymer chains | 1 |
Total formula weight | 24344.20 |
Authors | Bensen, D.C.,Akers-Rodriguez, S.,Lam, T.,Tari, L.W. (deposition date: 2013-04-12, release date: 2014-01-15, Last modification date: 2023-09-20) |
Primary citation | Tari, L.W.,Bensen, D.C.,Finn, J. A new class of type IIA topoisomerase inhibitors with broad-spectrum antibacterial activity To be Published, |
Experimental method | X-RAY DIFFRACTION (1.3 Å) |
Structure validation
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