4K31
Crystal structure of apramycin bound to the leishmanial rRNA A-site
Summary for 4K31
Entry DOI | 10.2210/pdb4k31/pdb |
Related | 4K32 |
Descriptor | RNA (5'-R(*UP*UP*GP*CP*GP*UP*CP*GP*UP*UP*CP*CP*GP*GP*AP*AP*AP*AP*GP*UP*CP*GP*C)-3'), APRAMYCIN (3 entities in total) |
Functional Keywords | rrna duplex, ribosomal a-site, aminoglycoside, ribosome, rna, rna-antibiotic complex, rna/antibiotic |
Biological source | Leishmania |
Total number of polymer chains | 2 |
Total formula weight | 16871.09 |
Authors | Shalev, M.,Kondo, J.,Adir, N.,Baasov, T. (deposition date: 2013-04-10, release date: 2013-07-31, Last modification date: 2023-09-20) |
Primary citation | Shalev, M.,Kondo, J.,Kopelyanskiy, D.,Jaffe, C.L.,Adir, N.,Baasov, T. Identification of the molecular attributes required for aminoglycoside activity against Leishmania. Proc.Natl.Acad.Sci.USA, 110:13333-13338, 2013 Cited by PubMed: 23898171DOI: 10.1073/pnas.1307365110 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.415 Å) |
Structure validation
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