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4JQ4

AKR1C2 complex with indomethacin

Summary for 4JQ4
Entry DOI10.2210/pdb4jq4/pdb
Related4JQ1 4JQ2 4JQ3 4JQA 4JTQ 4JTR
DescriptorAldo-keto reductase family 1 member C2, INDOMETHACIN, NADP NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ... (7 entities in total)
Functional Keywordsoxidoreductase-oxidoreductase inhibitor complex, oxidoreductase/oxidoreductase inhibitor
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm : P52895
Total number of polymer chains2
Total formula weight78534.66
Authors
Yosaatmadja, Y.,Flanagan, J.U.,Squire, C.J. (deposition date: 2013-03-19, release date: 2014-04-02, Last modification date: 2024-04-03)
Primary citationYosaatmadja, Y.,Flanagan, J.U.,Squire, C.J.
Structural basis of NSAID selectivity for the aldo-keto reductase 1C family
To be Published,
Experimental method
X-RAY DIFFRACTION (1.52 Å)
Structure validation

218853

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