4JL9
Crystal structure of mouse TBK1 bound to BX795
Summary for 4JL9
Entry DOI | 10.2210/pdb4jl9/pdb |
Descriptor | Serine/threonine-protein kinase TBK1, N-(3-{[5-iodo-4-({3-[(thiophen-2-ylcarbonyl)amino]propyl}amino)pyrimidin-2-yl]amino}phenyl)pyrrolidine-1-carboxamide (2 entities in total) |
Functional Keywords | protein kinase, kinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Mus musculus (mouse) |
Total number of polymer chains | 1 |
Total formula weight | 76281.84 |
Authors | |
Primary citation | Shu, C.,Sankaran, B.,Chaton, C.T.,Herr, A.B.,Mishra, A.,Peng, J.,Li, P. Structural Insights into the Functions of TBK1 in Innate Antimicrobial Immunity. Structure, 21:1137-1148, 2013 Cited by PubMed: 23746807DOI: 10.1016/j.str.2013.04.025 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.0999 Å) |
Structure validation
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