4JIN
X-ray crystal structure of Archaeoglobus fulgidus Rio1 bound to (2E)-N-benzyl-2-cyano-3-(pyridine-4-yl)acrylamide (WP1086)
Summary for 4JIN
Entry DOI | 10.2210/pdb4jin/pdb |
Related | 1ZP9 1ZTF |
Descriptor | RIO-type serine/threonine-protein kinase Rio1, (2E)-N-benzyl-2-cyano-3-(pyridin-4-yl)prop-2-enamide (3 entities in total) |
Functional Keywords | protein kinase, ribosome biogenesis, pre-40s, autophosphorylation, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Archaeoglobus fulgidus |
Total number of polymer chains | 1 |
Total formula weight | 30400.95 |
Authors | Mielecki, M.,Krawiec, K.,Kiburu, I.,Grzelak, K.,Wlodzimierz, Z.,Kierdaszuk, B.,Kowa, K.,Fokt, I.,Szymanski, S.,Piotr, S.,Szeja, W.,Priebe, W.,Lesyng, B.,LaRonde-LeBlanc, N. (deposition date: 2013-03-06, release date: 2013-04-24, Last modification date: 2023-09-20) |
Primary citation | Mielecki, M.,Krawiec, K.,Kiburu, I.,Grzelak, K.,Zagorski, W.,Kierdaszuk, B.,Kowa, K.,Fokt, I.,Szymanski, S.,Swierk, P.,Szeja, W.,Priebe, W.,Lesyng, B.,Laronde-Leblanc, N. Development of novel molecular probes of the Rio1 atypical protein kinase. Biochim.Biophys.Acta, 1834:1292-1301, 2013 Cited by PubMed: 23523885DOI: 10.1016/j.bbapap.2013.03.012 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.095 Å) |
Structure validation
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