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4J4N

Crystal structure of FK506 binding domain of plasmodium falciparum FKBP35 in complex with D44

Summary for 4J4N
Entry DOI10.2210/pdb4j4n/pdb
Related2OFN 2VN1 4J4O
DescriptorFK506-binding protein (FKBP)-type peptidyl-propyl isomerase, N-(2-ethylphenyl)-2-(3H-imidazo[4,5-b]pyridin-2-ylsulfanyl)acetamide (3 entities in total)
Functional Keywordsd44, fkbp35, fk506 binding, isomerase-isomerase inhibitor complex, isomerase/isomerase inhibitor
Biological sourcePlasmodium falciparum
Total number of polymer chains3
Total formula weight44531.43
Authors
Sreekanth, R.,Harikishore, A.,Yoon, H.S. (deposition date: 2013-02-07, release date: 2013-09-11, Last modification date: 2023-11-08)
Primary citationHarikishore, A.,Niang, M.,Rajan, S.,Preiser, P.R.,Yoon, H.S.
Small molecule Plasmodium FKBP35 inhibitor as a potential antimalaria agent.
Sci Rep, 3:2501-2501, 2013
Cited by
PubMed: 23974147
DOI: 10.1038/srep02501
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.75 Å)
Structure validation

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