4GUB

Casein Kinase II bound to Inhibitor

Summary for 4GUB

• Entry DOI: 10.2210/pdb4gub/pdb
• Related: 3U4U
• Descriptor: Casein kinase II subunit alpha, N-[5-({3-cyano-7-[(1-methyl-1H-imidazol-4-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl}amino)-2-methylphenyl]acetamide, CHLORIDE ION, ... (4 entities in total)
• Functional Keywords: kinase, transferase, cytosol, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 40315.37

Authors

Larsen, N.A.,Dowling, J.E. (deposition date: 2012-08-29, release date: 2013-09-25, Last modification date: 2024-02-28)

• Primary citation: Dowling, J.E.,Larsen, N.A.; Potent and selective inhibitors of CK2 kinase.; To be Published,

Experimental method

X-RAY DIFFRACTION (2.2 Å)