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4DON

Brd4 Bromodomain 1 complex with a fragment 3,4-Dihydro-3-methyl-2(1H)-quinazolinon

Summary for 4DON
Entry DOI10.2210/pdb4don/pdb
DescriptorBromodomain-containing protein 4, 3-methyl-3,4-dihydroquinazolin-2(1H)-one (3 entities in total)
Functional Keywordsbrd4, bromodomain, four alpha helices, signaling protein
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight17387.94
Authors
Xiong, B.,Cao, D.Y.,Chen, W.Y.,Chen, T.T.,Xu, Y.C.,Shen, J.K. (deposition date: 2012-02-09, release date: 2013-02-13, Last modification date: 2024-03-20)
Primary citationXiong, B.,Cao, D.Y.,Chen, W.Y.,Chen, T.T.,Xu, Y.C.,Shen, J.K.
Brd4 Bromodomain 1 complex with a fragment 3,4-Dihydro-3-methyl-2(1H)-quinazolinon
To be Published,
Experimental method
X-RAY DIFFRACTION (1.52 Å)
Structure validation

221051

数据于2024-06-12公开中

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