4CA8
Drosophila Angiotensin converting enzyme (AnCE) in complex with a phosphinic tripeptide FII
4CA8 の概要
エントリーDOI | 10.2210/pdb4ca8/pdb |
関連するPDBエントリー | 4CA5 4CA6 4CA7 |
分子名称 | ANGIOTENSIN-CONVERTING ENZYME, beta-D-mannopyranose-(1-6)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, [(2S)-2-({3-[HYDROXYL(2-PHENYL-(1R)-1-{[(BENZYLOXY)[(2S)-2-({3-[HYDROXYL(2-PHENYL-(1R)-1-CARBONYL]-AMINO}ETHYL)PHOSPHINYL]-2-[(3-PHENYLISOXAZOL-5-YL)METHYL]-1-OXO-PROPYL}AMINO)-3-(4-HYDROXY-PHENYL), ... (7 entities in total) |
機能のキーワード | hydrolase, zinc metallopeptidase, inhibitor binding |
由来する生物種 | DROSOPHILA MELANOGASTER (FRUIT FLY) |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 71829.34 |
構造登録者 | Masuyer, G.,Akif, M.,Czarny, B.,Beau, F.,Schwager, S.L.U.,Sturrock, E.D.,Isaac, R.E.,Dive, V.,Acharya, K.R. (登録日: 2013-10-07, 公開日: 2013-12-11, 最終更新日: 2024-10-09) |
主引用文献 | Masuyer, G.,Akif, M.,Czarny, B.,Beau, F.,Schwager, S.L.,Sturrock, E.D.,Isaac, R.E.,Dive, V.,Acharya, K.R. Crystal Structures of Highly Specific Phosphinic Tripeptide Enantiomers in Complex with the Angiotensin-I Converting Enzyme. FEBS J., 281:943-, 2014 Cited by PubMed: 24289879DOI: 10.1111/FEBS.12660 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.99 Å) |
構造検証レポート
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