4ANS
Structure of L1196M,G1269A Double Mutant Anaplastic Lymphoma Kinase in Complex with Crizotinib
Summary for 4ANS
Entry DOI | 10.2210/pdb4ans/pdb |
Related | 4ANL 4ANQ 4AOI |
Descriptor | ALK TYROSINE KINASE RECEPTOR, 3-[(1R)-1-(2,6-dichloro-3-fluorophenyl)ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)pyridin-2-amine (3 entities in total) |
Functional Keywords | transferase |
Biological source | HOMO SAPIENS (HUMAN) |
Total number of polymer chains | 1 |
Total formula weight | 39078.53 |
Authors | McTigue, M.,Deng, Y.,Liu, W.,Brooun, A. (deposition date: 2012-03-22, release date: 2013-03-27, Last modification date: 2023-12-20) |
Primary citation | Mctigue, M.,Deng, Y.,Liu, W.,Brooun, A. Structure of L1196M,G1269A Double Mutant Anaplastic Lymphoma Kinase in Complex with Crizotinib To be Published, |
Experimental method | X-RAY DIFFRACTION (1.85 Å) |
Structure validation
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