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4XSZ

Crystal structure of CBR 9393 bound to Escherichia coli RNA polymerase holoenzyme

Summary for 4XSZ
Entry DOI10.2210/pdb4xsz/pdb
Related4XSX 4XSY
DescriptorDNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, DNA-directed RNA polymerase subunit beta', ... (8 entities in total)
Functional Keywordsbacterial rna polymerase antibiotic complex, transcription-antibiotic complex, transcription/antibiotic
Biological sourceEscherichia coli (strain K12)
More
Cellular locationCytoplasm : P00579
Total number of polymer chains12
Total formula weight860518.55
Authors
Bae, B.,Darst, S.A. (deposition date: 2015-01-22, release date: 2015-07-22, Last modification date: 2023-09-27)
Primary citationBae, B.,Nayak, D.,Ray, A.,Mustaev, A.,Landick, R.,Darst, S.A.
CBR antimicrobials inhibit RNA polymerase via at least two bridge-helix cap-mediated effects on nucleotide addition.
Proc.Natl.Acad.Sci.USA, 112:E4178-E4187, 2015
Cited by
PubMed: 26195788
DOI: 10.1073/pnas.1502368112
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3.683 Å)
Structure validation

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