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4U7H

Oxidized quinone reductase 2 in complex with CK2 inhibitor DMAT

Summary for 4U7H
Entry DOI10.2210/pdb4u7h/pdb
Related4U7F 4U7G
DescriptorRibosyldihydronicotinamide dehydrogenase [quinone], ZINC ION, FLAVIN-ADENINE DINUCLEOTIDE, ... (5 entities in total)
Functional Keywordsreduced quinone reductase 2, dmat, oxidoreductase-inhibitor complex, oxidoreductase/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationCytoplasm: P16083
Total number of polymer chains2
Total formula weight54354.17
Authors
Leung, K.K.,Shilton, B.H. (deposition date: 2014-07-30, release date: 2015-02-11, Last modification date: 2023-12-27)
Primary citationLeung, K.K.,Shilton, B.H.
Quinone Reductase 2 Is an Adventitious Target of Protein Kinase CK2 Inhibitors TBBz (TBI) and DMAT.
Biochemistry, 54:47-59, 2015
Cited by
PubMed: 25379648
DOI: 10.1021/bi500959t
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.48 Å)
Structure validation

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