4TS8

Crystal structure of the bromodomain of human CREBBP in complex with XZ08

Summary for 4TS8

• Entry DOI: 10.2210/pdb4ts8/pdb
• Descriptor: CREB-binding protein, 1,2-ETHANEDIOL, 4-(1-acetyl-1H-indol-3-yl)-5-methyl-1,2-dihydro-3H-pyrazol-3-one, ... (4 entities in total)
• Functional Keywords: transcription, inhibitor, transferase
• Biological source: Homo sapiens (Human)
• Cellular location: Cytoplasm: Q92793
• Total number of polymer chains: 1
• Total formula weight: 14602.76

Authors

Dong, J.,Gartenmann, L.,Spiliotopoulos, D.,Caflisch, A. (deposition date: 2014-06-18, release date: 2015-07-01, Last modification date: 2023-12-20)

• Primary citation: Dong, J.,Gartenmann, L.,Spiliotopoulos, D.,Caflisch, A.; Crystal structure of the bromodomain of human CREBBP in complex with XZ08; To Be Published,

Experimental method

X-RAY DIFFRACTION (2 Å)