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4TS8

Crystal structure of the bromodomain of human CREBBP in complex with XZ08

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue EDO A 1201
ChainResidue
AASP1155
ALEU1159
AASN1162
AHOH1324
AHOH1325

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 1202
ChainResidue
ALEU1120
ATRP1165
AHOH1301
AHOH1306

site_idAC3
Number of Residues8
Detailsbinding site for residue XZ8 A 1203
ChainResidue
APRO1110
AILE1122
AASN1168
AVAL1174
AHOH1301
AHOH1305
AHOH1372
AHOH1378

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

224931

PDB entries from 2024-09-11

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