4F21
Crystal structure of carboxylesterase/phospholipase family protein from Francisella tularensis
Summary for 4F21
Entry DOI | 10.2210/pdb4f21/pdb |
Descriptor | Carboxylesterase/phospholipase family protein, N-((1R,2S)-2-allyl-4-oxocyclobutyl)-4-methylbenzenesulfonamide, bound form (3 entities in total) |
Functional Keywords | structural genomics, niaid, national institute of allergy and infectious diseases, center for structural genomics of infectious diseases, csgid, carboxylesterase, phospholipase, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
Biological source | Francisella tularensis subsp. tularensis |
Total number of polymer chains | 8 |
Total formula weight | 219795.92 |
Authors | Filippova, E.V.,Minasov, G.,Kuhn, M.,Wawrzak, Z.,Shuvalova, L.,Dubrovska, I.,Winsor, J.R.,Kiryukhina, O.,Becker, D.P.,Armoush, N.,Anderson, W.F.,Center for Structural Genomics of Infectious Diseases (CSGID) (deposition date: 2012-05-07, release date: 2012-08-29, Last modification date: 2023-09-13) |
Primary citation | Filippova, E.V.,Weston, L.A.,Kuhn, M.L.,Geissler, B.,Gehring, A.M.,Armoush, N.,Adkins, C.T.,Minasov, G.,Dubrovska, I.,Shuvalova, L.,Winsor, J.R.,Lavis, L.D.,Satchell, K.J.,Becker, D.P.,Anderson, W.F.,Johnson, R.J. Large scale structural rearrangement of a serine hydrolase from Francisella tularensis facilitates catalysis. J.Biol.Chem., 288:10522-10535, 2013 Cited by PubMed: 23430251DOI: 10.1074/jbc.M112.446625 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.5 Å) |
Structure validation
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