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4D5H

Focal Adhesion Kinase catalytic domain

Summary for 4D5H
Entry DOI10.2210/pdb4d5h/pdb
Related4D4R 4D4S 4D4V 4D4Y 4D55 4D58 4D5K
DescriptorFOCAL ADHESION KINASE 1, 6-methyl-5-{[3-(trifluoromethyl)phenyl]amino}-1,2,4-triazin-3(4H)-one, SULFATE ION, ... (4 entities in total)
Functional Keywordstransferase, kinase inhibitor, atp-binding, integrin signaling
Biological sourceGALLUS GALLUS (CHICKEN)
Total number of polymer chains2
Total formula weight64118.07
Authors
Le Coq, J.,Lin, A.,Lietha, D. (deposition date: 2014-11-05, release date: 2015-02-18, Last modification date: 2023-12-20)
Primary citationZhou, J.,Bronowska, A.,Le Coq, J.,Lietha, D.,Grater, F.
Allosteric Regulation of Focal Adhesion Kinase by Pip2 and ATP.
Biophys.J., 108:698-, 2015
Cited by
PubMed: 25650936
DOI: 10.1016/J.BPJ.2014.11.3454
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

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