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3WJ4

Crystal structure of PPARgamma ligand binding domain in complex with tributyltin

Summary for 3WJ4
Entry DOI10.2210/pdb3wj4/pdb
Related3WJ5
DescriptorPeroxisome proliferator-activated receptor gamma, tributylstannanyl (3 entities in total)
Functional Keywordsprotein-ligand complex, dna-binding, metal-binding, nucleus, receptor, transcription
Biological sourceHomo sapiens (human)
Cellular locationNucleus: P37231
Total number of polymer chains2
Total formula weight63397.04
Authors
Harada, S.,Hiromori, Y.,Fukakusa, S.,Kawahara, K.,Nakamura, S.,Noda, M.,Uchiyama, S.,Fukui, K.,Nishikawa, J.,Nagase, H.,Kobayashi, Y.,Ohkubo, T.,Yoshida, T.,Nakanishi, T. (deposition date: 2013-10-04, release date: 2014-10-15, Last modification date: 2024-03-20)
Primary citationHarada, S.,Hiromori, Y.,Fukakusa, S.,Kawahara, K.,Nakamura, S.,Noda, M.,Uchiyama, S.,Fukui, K.,Nishikawa, J.,Nagase, H.,Kobayashi, Y.,Ohkubo, T.,Yoshida, T.,Nakanishi, T.
Structural basis for PPARgamma transactivation by endocrine disrupting organotin compounds
To be Published,
Experimental method
X-RAY DIFFRACTION (1.95 Å)
Structure validation

217705

건을2024-03-27부터공개중

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