3UZP
crystal structure of ck1d with PF670462 from P21 crystal form
Summary for 3UZP
| Entry DOI | 10.2210/pdb3uzp/pdb |
| Related | 1CKI 3UYS 3UYT |
| Descriptor | Casein kinase I isoform delta, 4-[1-cyclohexyl-4-(4-fluorophenyl)-1H-imidazol-5-yl]pyrimidin-2-amine (3 entities in total) |
| Functional Keywords | ck1d, kinase, inhibitor, pf670462, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
| Biological source | Homo sapiens (human) |
| Cellular location | Cytoplasm: P48730 |
| Total number of polymer chains | 2 |
| Total formula weight | 69376.11 |
| Authors | Huang, X. (deposition date: 2011-12-07, release date: 2012-01-11, Last modification date: 2024-02-28) |
| Primary citation | Long, A.,Zhao, H.,Huang, X. Structural basis for the interaction between casein kinase 1 delta and a potent and selective inhibitor. J.Med.Chem., 55:956-960, 2012 Cited by PubMed: 22168824DOI: 10.1021/jm201387s PDB entries with the same primary citation |
| Experimental method | X-RAY DIFFRACTION (1.94 Å) |
Structure validation
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