3UVR

Human p38 MAP Kinase in Complex with KM064

Summary for 3UVR

• Entry DOI: 10.2210/pdb3uvr/pdb
• Related: 3QUD 3QUE 3UVP 3UVQ 3UVS
• Descriptor: Mitogen-activated protein kinase 14, 1-[3-tert-butyl-1-(4-methylphenyl)-1H-pyrazol-5-yl]-3-{3-[(5-oxo-6,7,8,9-tetrahydro-5H-benzo[7]annulen-2-yl)amino]phenyl}urea, octyl beta-D-glucopyranoside, ... (4 entities in total)
• Functional Keywords: protein kinase, selective p38 inhibitor, sar, annulen derivative, pyrazolo urea, transferase-transferase inhibitor complex, transferase/transferase inhibitor
• Biological source: Homo sapiens (human)
• Total number of polymer chains: 1
• Total formula weight: 42375.45

Authors

Richters, A.,Mayer-Wrangowski, S.C.,Gruetter, C.,Rauh, D. (deposition date: 2011-11-30, release date: 2012-12-19, Last modification date: 2023-11-08)

• Primary citation: ; ,

Experimental method

X-RAY DIFFRACTION (2.1 Å)