3UH2
Tankyrase-1 in complexed with PJ34
Summary for 3UH2
Entry DOI | 10.2210/pdb3uh2/pdb |
Related | 3UH4 |
Descriptor | Tankyrase-1, ZINC ION, N~2~,N~2~-DIMETHYL-N~1~-(6-OXO-5,6-DIHYDROPHENANTHRIDIN-2-YL)GLYCINAMIDE, ... (5 entities in total) |
Functional Keywords | transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm: O95271 |
Total number of polymer chains | 2 |
Total formula weight | 52611.90 |
Authors | Kirby, C.A.,Stams, T. (deposition date: 2011-11-03, release date: 2012-02-15, Last modification date: 2023-09-13) |
Primary citation | Kirby, C.A.,Cheung, A.,Fazal, A.,Shultz, M.D.,Stams, T. Structure of human tankyrase 1 in complex with small-molecule inhibitors PJ34 and XAV939. Acta Crystallogr.,Sect.F, 68:115-118, 2012 Cited by PubMed: 22297980DOI: 10.1107/S1744309111051219 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2 Å) |
Structure validation
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