3SA0
Complex of ERK2 with norathyriol
Summary for 3SA0
Entry DOI | 10.2210/pdb3sa0/pdb |
Related | 1TVO |
Descriptor | Mitogen-activated protein kinase 1, norathyriol, SULFATE ION, ... (4 entities in total) |
Functional Keywords | norathyriol complex, signal-regulated kinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Nucleus: P28482 |
Total number of polymer chains | 1 |
Total formula weight | 42029.27 |
Authors | Kurinov, I.,Malakhova, M. (deposition date: 2011-06-02, release date: 2011-12-14, Last modification date: 2023-09-13) |
Primary citation | Li, J.,Malakhova, M.,Mottamal, M.,Reddy, K.,Kurinov, I.,Carper, A.,Langfald, A.,Oi, N.,Kim, M.O.,Zhu, F.,Sosa, C.P.,Zhou, K.,Bode, A.M.,Dong, Z. Norathyriol Suppresses Skin Cancers Induced by Solar Ultraviolet Radiation by Targeting ERK Kinases. Cancer Res., 72:260-270, 2012 Cited by PubMed: 22084399DOI: 10.1158/0008-5472.CAN-11-2596 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.5947 Å) |
Structure validation
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