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3RDH

X-ray induced covalent inhibition of 14-3-3

Summary for 3RDH
Entry DOI10.2210/pdb3rdh/pdb
Descriptor14-3-3 protein zeta/delta, 4-[(E)-{4-formyl-5-hydroxy-6-methyl-3-[(phosphonooxy)methyl]pyridin-2-yl}diazenyl]benzoic acid, NICKEL (II) ION, ... (4 entities in total)
Functional Keywordsphosphoser/thr-mimetic agent, phosphoserine/threonine-recognition protein, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (human)
Cellular locationCytoplasm: P63104
Total number of polymer chains4
Total formula weight114053.29
Authors
Horton, J.R.,Upadhyay, A.K.,Fu, H.,Cheng, X. (deposition date: 2011-04-01, release date: 2011-09-28, Last modification date: 2023-09-13)
Primary citationZhao, J.,Du, Y.,Horton, J.R.,Upadhyay, A.K.,Lou, B.,Bai, Y.,Zhang, X.,Du, L.,Li, M.,Wang, B.,Zhang, L.,Barbieri, J.T.,Khuri, F.R.,Cheng, X.,Fu, H.
Discovery and structural characterization of a small molecule 14-3-3 protein-protein interaction inhibitor.
Proc.Natl.Acad.Sci.USA, 108:16212-16216, 2011
Cited by
PubMed: 21908710
DOI: 10.1073/pnas.1100012108
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.39 Å)
Structure validation

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