3QBN
Structure of Human Aurora A in Complex with a diaminopyrimidine
Summary for 3QBN
Entry DOI | 10.2210/pdb3qbn/pdb |
Descriptor | Serine/threonine-protein kinase 6, 5-chloro-N~4~-cyclopropyl-N~2~-[4-(2-methoxyethoxy)phenyl]pyrimidine-2,4-diamine (2 entities in total) |
Functional Keywords | kinase domain, diaminopyrimidine, transferase-transferase inhibitor complex, transferase/transferase inhibitor |
Biological source | Homo sapiens (human) |
Cellular location | Cytoplasm, cytoskeleton, centrosome: O14965 |
Total number of polymer chains | 1 |
Total formula weight | 32837.01 |
Authors | Gruetter, C.,Simard, J.R.,Rauh, D. (deposition date: 2011-01-13, release date: 2012-01-18, Last modification date: 2023-09-13) |
Primary citation | Tueckmantel, S.,Greul, J.N.,Janning, P.,Brockmeyer, A.,Gruetter, C.,Simard, J.R.,Gutbrod, O.,Beck, M.E.,Tietjen, K.,Rauh, D.,Schreier, P.H. Identification of Ustilago maydis Aurora kinase as a novel antifungal target. Acs Chem.Biol., 6:926-933, 2011 Cited by PubMed: 21671622DOI: 10.1021/cb200112y PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (3.5 Å) |
Structure validation
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