3HMI
The crystal structure of human ABL2 in complex with 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE
3HMI の概要
エントリーDOI | 10.2210/pdb3hmi/pdb |
関連するPDBエントリー | 3GVU |
分子名称 | Tyrosine-protein kinase ABL2, 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE (3 entities in total) |
機能のキーワード | tyrosine kinase, abl, abl2, abelson murine leukemia viral oncogene, atp-binding, cell adhesion, cytoskeleton, kinase, lipoprotein, magnesium, manganese, metal-binding, myristate, nucleotide-binding, phosphoprotein, sh2 domain, sh3 domain, transferase, tyrosine-protein kinase, structural genomics, structural genomics consortium, sgc |
由来する生物種 | Homo sapiens (human) |
細胞内の位置 | Cytoplasm, cytoskeleton: P42684 |
タンパク質・核酸の鎖数 | 1 |
化学式量合計 | 33968.79 |
構造登録者 | Ugochukwu, E.,Salah, E.,Barr, A.,Mahajan, P.,Shrestha, B.,Savitsky, P.,Chaikuad, A.,Allerston, C.,von Delft, F.,Bountra, C.,Arrowsmith, C.H.,Weigelt, J.,Edwards, A.,Knapp, S.,Structural Genomics Consortium (SGC) (登録日: 2009-05-29, 公開日: 2009-07-07, 最終更新日: 2023-11-01) |
主引用文献 | Ugochukwu, E.,Salah, E.,Barr, A.,Mahajan, P.,Shrestha, B.,Savitsky, P.,Chaikuad, A.,Allerston, C.,von Delft, F.,Knapp, S. The crystal structure of human ABL2 in complex with 5-AMINO-3-{[4-(AMINOSULFONYL)PHENYL]AMINO}-N-(2,6-DIFLUOROPHENYL)-1H-1,2,4-TRIAZOLE-1-CARBOTHIOAMIDE To be Published, |
実験手法 | X-RAY DIFFRACTION (1.65 Å) |
構造検証レポート
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