3HIW
Crystal structure of Saporin-L1 in complex with the cyclic tetranucleotide inhibitor, a transition state analogue
3HIW の概要
エントリーDOI | 10.2210/pdb3hiw/pdb |
関連するPDBエントリー | 3HIO 3HIQ 3HIS 3HIT 3HIV |
分子名称 | Vacuolar saporin, 9,9'-{(2R,3R,3aR,5S,7aR,9R,10R,10aR,12S,23R,25aR,27R,28R,28aR,30S,32aR,35aR,37S,39aR)-9-(6-amino-9H-purin-9-yl)-34-[(4-amino-5H-pyrrolo[3,2-d]pyrimidin-7-yl)methyl]-5,12,23,30,37-pentahydroxy-3,10,28-trimethoxy-5,12,23,30,37-pentaoxidotetracosahydro-2H,7H,25H-trifuro[3,2-f:3',2'-l:3'',2''-x]pyrrolo[3,4-r][1,3,5,9,11,15,17,21,23,27,29,2,4,10,16,22,28]undecaoxazapentaphosphacyclopentatriacontine-2,27-diyl}bis(2-amino-3,9-dihydro-6H-purin-6-one) (3 entities in total) |
機能のキーワード | transition state, ribosome inactivating proteins, rips, hydrolase, plant defense, protein synthesis inhibitor, toxin, hydrolase-hydrolase inhibitor complex, hydrolase/hydrolase inhibitor |
由来する生物種 | Saponaria officinalis (Common soapwort) |
タンパク質・核酸の鎖数 | 2 |
化学式量合計 | 60731.76 |
構造登録者 | |
主引用文献 | Ho, M.C.,Sturm, M.B.,Almo, S.C.,Schramm, V.L. Transition state analogues in structures of ricin and saporin ribosome-inactivating proteins. Proc.Natl.Acad.Sci.USA, 106:20276-20281, 2009 Cited by PubMed: 19920175DOI: 10.1073/pnas.0911606106 主引用文献が同じPDBエントリー |
実験手法 | X-RAY DIFFRACTION (1.8 Å) |
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