3G15
Crystal structure of human choline kinase alpha in complex with hemicholinium-3 and ADP
Replaces: 3F2SSummary for 3G15
Entry DOI | 10.2210/pdb3g15/pdb |
Related | 3F2S |
Descriptor | Choline kinase alpha, ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, ... (7 entities in total) |
Functional Keywords | non-protein kinase, choline kinase, structural genomics consortium, sgc, hemicholinium-3, kinase, transferase |
Biological source | Homo sapiens (human) |
Total number of polymer chains | 2 |
Total formula weight | 95685.78 |
Authors | Hong, B.S.,Tempel, W.,Rabeh, W.M.,MacKenzie, F.,Arrowsmith, C.H.,Edwards, A.M.,Bountra, C.,Weigelt, J.,Bochkarev, A.,Park, H.W.,Structural Genomics Consortium (SGC) (deposition date: 2009-01-29, release date: 2009-02-10, Last modification date: 2023-09-06) |
Primary citation | Hong, B.S.,Allali-Hassani, A.,Tempel, W.,Finerty, P.J.,Mackenzie, F.,Dimov, S.,Vedadi, M.,Park, H.W. Crystal structures of human choline kinase isoforms in complex with hemicholinium-3: single amino acid near the active site influences inhibitor sensitivity. J.Biol.Chem., 285:16330-16340, 2010 Cited by PubMed: 20299452DOI: 10.1074/jbc.M109.039024 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.7 Å) |
Structure validation
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