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3FSI

Crystal structure of a trypanocidal 4,4'-Bis(imidazolinylamino)diphenylamine bound to DNA

Summary for 3FSI
Entry DOI10.2210/pdb3fsi/pdb
DescriptorReverse transcriptase domain, 5'-D(*CP*TP*TP*AP*AP*TP*TP*C)-3', 5'-D(P*GP*AP*AP*TP*TP*AP*AP*G)-3', ... (6 entities in total)
Functional Keywordstransferase/dna mmlv rt, protein-dna complex, drug-dna complex, cd27, antitrypanosomal, dna integration, dna recombination, nucleotidyltransferase, transferase, transferase-dna complex, transferase/dna
Biological sourceMoloney murine leukemia virus (Virus)
Cellular locationGag-Pol polyprotein: Host cell membrane ; Lipid-anchor . Matrix protein p15: Virion . Capsid protein p30: Virion . Nucleocapsid protein p10: Virion : P03355
Total number of polymer chains3
Total formula weight34416.17
Authors
Glass, L.S.,Georgiadis, M.M.,Goodwin, K.D. (deposition date: 2009-01-09, release date: 2009-05-19, Last modification date: 2023-09-06)
Primary citationGlass, L.S.,Nguyen, B.,Goodwin, K.D.,Dardonville, C.,Wilson, W.D.,Long, E.C.,Georgiadis, M.M.
Crystal structure of a trypanocidal 4,4'-bis(imidazolinylamino)diphenylamine bound to DNA.
Biochemistry, 48:5943-5952, 2009
Cited by
PubMed: 19405506
DOI: 10.1021/bi900204w
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

217705

數據於2024-03-27公開中

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