3FSI
Crystal structure of a trypanocidal 4,4'-Bis(imidazolinylamino)diphenylamine bound to DNA
Summary for 3FSI
Entry DOI | 10.2210/pdb3fsi/pdb |
Descriptor | Reverse transcriptase domain, 5'-D(*CP*TP*TP*AP*AP*TP*TP*C)-3', 5'-D(P*GP*AP*AP*TP*TP*AP*AP*G)-3', ... (6 entities in total) |
Functional Keywords | transferase/dna mmlv rt, protein-dna complex, drug-dna complex, cd27, antitrypanosomal, dna integration, dna recombination, nucleotidyltransferase, transferase, transferase-dna complex, transferase/dna |
Biological source | Moloney murine leukemia virus (Virus) |
Cellular location | Gag-Pol polyprotein: Host cell membrane ; Lipid-anchor . Matrix protein p15: Virion . Capsid protein p30: Virion . Nucleocapsid protein p10: Virion : P03355 |
Total number of polymer chains | 3 |
Total formula weight | 34416.17 |
Authors | Glass, L.S.,Georgiadis, M.M.,Goodwin, K.D. (deposition date: 2009-01-09, release date: 2009-05-19, Last modification date: 2023-09-06) |
Primary citation | Glass, L.S.,Nguyen, B.,Goodwin, K.D.,Dardonville, C.,Wilson, W.D.,Long, E.C.,Georgiadis, M.M. Crystal structure of a trypanocidal 4,4'-bis(imidazolinylamino)diphenylamine bound to DNA. Biochemistry, 48:5943-5952, 2009 Cited by PubMed: 19405506DOI: 10.1021/bi900204w PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.75 Å) |
Structure validation
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