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3F2N

Crystal Structure of Human Haspin with an Imidazo-pyridazine ligand

Summary for 3F2N
Entry DOI10.2210/pdb3f2n/pdb
DescriptorSerine/threonine-protein kinase haspin, (2S)-2-{[3-(3-aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino}-3-methylbutan-1-ol, PHOSPHATE ION, ... (5 entities in total)
Functional Keywordshaspin, germ cell associated 2, haploid germ cell specific nuclear protein kinase, atp-binding, cell cycle, chromatin regulator, kinase, magnesium, nucleotide-binding, nucleus, phosphoprotein, serine/threonine-protein kinase, transferase, structural genomics, structural genomics consortium, sgc
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: Q8TF76
Total number of polymer chains1
Total formula weight41428.18
Authors
Primary citationFilippakopoulos, P.,Eswaran, J.,Keates, T.,Burgess-Brown, N.,Fedorov, O.,Yue, W.W.,Murray, J.W.,Pike, A.C.W.,Von Delft, F.,Arrowsmith, C.H.,Edwards, A.M.,Weigelt, J.,Bountra, C.,Knapp, S.
Crystal Structure of Human Haspin with an Imidazo-pyridazine ligand
To be Published,
Experimental method
X-RAY DIFFRACTION (1.8 Å)
Structure validation

217705

건을2024-03-27부터공개중

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